SCHEMBL22112367

SCHEMBL22112367

Oc1cccc(C[C@H]2CCC=C(N3CCC3)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
MGLL Q99685 1/20 0.39
OPRM1 P35372 10/20 0.38
OPRK1 P41145 10/20 0.38
OPRD1 P41143 9/20 0.38
CYP19A1 P11511 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2967942 0.74 OPRM1 (0.59) ESR1ESR2OPRM1OPRK1OPRD1
SCHEMBL22112096 0.74 ESR1 (0.43) ESR1ESR2OPRM1OPRK1OPRD1
SCHEMBL14143096 0.73 OPRM1 (0.60) ESR1ESR2OPRM1OPRK1OPRD1
SCHEMBL6932394 0.69 CCR3 (0.44) MGLL
SCHEMBL30503933 0.69 OPRM1 (0.51) ESR1ESR2MGLLOPRM1OPRK1
SCHEMBL12230207 0.68 CCR3 (0.50) MGLL
SCHEMBL27785492 0.68 GBA1 (0.62) ESR1ESR2OPRM1OPRK1OPRD1
SCHEMBL22112048 0.66 ESR2 (0.49) ESR1ESR2MGLLOPRM1OPRK1
SCHEMBL7053655 0.65 KCNH2 (0.43) MGLLDRD2DRD3
SCHEMBL28052784 0.65 GRIN2D (0.53) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020120539-A1 NEW PYRROLIDINE-2-CARBOXYLIC ACID DERIVATIVES FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-06-18 WO disclosed