SCHEMBL22115151

SCHEMBL22115151

CC(C)(C)OC(=O)N1CCC(C)(C(=O)NS(=O)(=O)c2ccc(Cl)s2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 8/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44
P2RY12 Q9H244 2/20 0.43
MMP13 P45452 5/20 0.42
MMP1 P03956 2/20 0.42
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NTRK1 P04629 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4100013 0.81 STS (0.69) STSP2RY12MMP13MMP1MAPT
SCHEMBL1168528 0.80 STS (0.44) STSPSEN1PSEN2APH1BNCSTN
SCHEMBL22089492 0.78 STS (0.57) STSPSEN1PSEN2APH1BNCSTN
SCHEMBL22115155 0.78 STS (0.40) STSCYP2C9MMP13MAPTNTRK1
SCHEMBL22115699 0.77 CYP1A2 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL22089522 0.77 STS (0.55) STSCYP3A4MMP13
SCHEMBL28079459 0.75 PSEN1 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL22115318 0.73 STS (0.55) STSCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1563895 0.73 ALDH1A1 (0.54) STSPSEN1PSEN2APH1BNCSTN
SCHEMBL1668225 0.72 MEN1 (0.44) STSMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111303146-A 3-cyanopyridine compound, pharmaceutical composition containing same, preparation method and application thereof 中国科学院上海药物研究所 2020-06-19 CN disclosed
WO-2020119590-A1 3-CYANOPYRIDINE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, PREPARATION METHOD THEREFOR, AND USES THEREOF. 中国科学院上海药物研究所 2020-06-18 WO disclosed