SCHEMBL22115652

SCHEMBL22115652

CC(C)(C)OC(=O)N1CCC(C(=O)NSCc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
STS P08842 6/20 0.53
PTPN2 P17706 1/20 0.50
PTPN1 P18031 1/20 0.50
PTPN6 P29350 1/20 0.50
KMT2A Q03164 1/20 0.49
MAPT P10636 1/20 0.49
EPHX2 P34913 1/20 0.48
TGFBR1 P36897 1/20 0.47
GPR119 Q8TDV5 1/20 0.46
TACR1 P25103 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ABL1 P00519 1/20 0.44
RIN1 Q13671 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PKM P14618 1/20 0.44
P2RY14 Q15391 1/20 0.44
MMP13 P45452 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22115171 0.87 STS (0.60) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL22115157 0.87 STS (0.64) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL22115696 0.82 STS (0.58) STSPTPN2PTPN1PTPN6GPR119
SCHEMBL22089514 0.80 STS (0.77) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL29716354 0.80 PTPN2 (0.77) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL311411 0.80 KMT2A (0.55) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL16112715 0.78 TGFBR1 (0.54) STSMAPTTGFBR1GPR119KDM4E
SCHEMBL20015404 0.78 MAOB (0.54) STSMAPTTGFBR1GPR119KDM4E
SCHEMBL4242260 0.77 HSD11B1 (0.62) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL22115170 0.77 STS (0.51) STSPTPN2PTPN1PTPN6GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020119590-A1 3-CYANOPYRIDINE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, PREPARATION METHOD THEREFOR, AND USES THEREOF. 中国科学院上海药物研究所 2020-06-18 WO disclosed