SCHEMBL22115706

SCHEMBL22115706

CC(C)(C)OC(=O)N1CCC(C(=O)NS(=O)(=O)Cc2ccc(C#N)cc2)CC1

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
STS P08842 10/20 0.77
GPR119 Q8TDV5 4/20 0.53
PTPN2 P17706 1/20 0.49
PTPN1 P18031 1/20 0.49
PTPN6 P29350 1/20 0.49
P2RY12 Q9H244 2/20 0.47
KMT2A Q03164 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28422888 0.95 STS (0.70) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL28422820 0.87 STS (0.80) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL22089512 0.87 STS (0.80) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL1970651 0.87 STS (1.00) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL22089514 0.85 STS (0.77) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL3929382 0.84 GPR119 (0.56) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL22089505 0.82 STS (0.90) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL28418216 0.82 STS (0.90) STSGPR119PTPN2PTPN1PTPN6
SCHEMBL22089534 0.81 STS (1.00) STSPTPN2PTPN1PTPN6KMT2A
SCHEMBL3146175 0.79 GPR119 (0.60) STSGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020119590-A1 3-CYANOPYRIDINE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, PREPARATION METHOD THEREFOR, AND USES THEREOF. 中国科学院上海药物研究所 2020-06-18 WO disclosed