SCHEMBL3929382

SCHEMBL3929382

CC(C)(C)OC(=O)N1CCC(C(=O)NCc2ccc(C#N)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.56
STS P08842 3/20 0.53
ALDH1A1 P00352 2/20 0.53
LMNA P02545 1/20 0.53
EPHX2 P34913 1/20 0.52
PTPN2 P17706 1/20 0.52
PTPN1 P18031 1/20 0.52
PTPN6 P29350 1/20 0.52
OGA O60502 1/20 0.49
NPSR1 Q6W5P4 2/20 0.49
KMT2A Q03164 2/20 0.48
CCR5 P51681 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK1 P28482 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984198 0.88 HDAC1 (0.54) GPR119ALDH1A1LMNAEPHX2NPSR1
SCHEMBL8266055 0.85 GPR119 (0.57) GPR119STSALDH1A1PTPN2PTPN1
SCHEMBL1668815 0.85 SMN1; SMN2 (0.52) GPR119ALDH1A1LMNAEPHX2NPSR1
SCHEMBL171943 0.85 STS (0.64) STSALDH1A1LMNAEPHX2PTPN2
SCHEMBL12804554 0.85 NPSR1 (0.68) GPR119STSALDH1A1LMNAEPHX2
SCHEMBL30924055 0.84 EPHX2 (0.58) GPR119STSALDH1A1EPHX2PTPN2
SCHEMBL27022355 0.84 ALDH1A1 (0.71) STSALDH1A1LMNAEPHX2KMT2A
SCHEMBL22115706 0.84 STS (0.77) GPR119STSPTPN2PTPN1PTPN6
SCHEMBL20116384 0.83 GPR119 (0.47) GPR119ALDH1A1LMNAEPHX2NPSR1
SCHEMBL13111226 0.83 ALDH1A1 (0.51) GPR119ALDH1A1LMNAEPHX2OGA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010480-A1 1-{2-[(DIPHENYL)AMINO]-ETHYL}-PIPERIDINE-4-CARBOXYLIC ACID BENZYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS CCR5 AGONISTS FOR THE TREATMENT OF IMMUNE AND INFLAMMATORY DISEASES EUROSCREEN S.A. (BE) 2009-01-22 WO disclosed