SCHEMBL22129208

SCHEMBL22129208

N#Cc1cc(N2C(=O)c3ccccc3C2=O)ccc1F

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.55
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
KCNH2 Q12809 1/20 0.44
SCN2A Q99250 5/20 0.43
PIM3 Q86V86 1/20 0.43
HIPK4 Q8NE63 1/20 0.43
NR1H3 Q13133 1/20 0.42
GRM1 Q13255 1/20 0.42
PGR P06401 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
PIM1 P11309 1/20 0.40
USP8 P40818 1/20 0.40
USP7 Q93009 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6689272 0.85 MEN1 (0.53) MEN1KMT2ASCN2APIM3HIPK4
SCHEMBL22163714 0.81 AR (0.48) ARDRD2DRD3KCNH2PGR
SCHEMBL14387538 0.78 GRM1 (0.44) MEN1KMT2ANR1H3GRM1PGR
SCHEMBL1633789 0.78 MEN1 (0.45) MEN1KMT2ASCN2APIM3HIPK4
SCHEMBL6676204 0.76 MEN1 (0.46) MEN1KMT2ASCN2APIM3HIPK4
SCHEMBL10999030 0.76 KMT2A (0.62) MEN1KMT2ASCN2APIM3HIPK4
SCHEMBL7360730 0.76 SCN2A (0.62) MEN1KMT2ASCN2APIM3HIPK4
SCHEMBL11520347 0.73 PGR (0.63) ARMEN1KMT2ASCN2ANR1H3
SCHEMBL5574945 0.72 POLB (0.49) ARMEN1KMT2ACA12CA1
SCHEMBL29870828 0.72 GRM5 (0.54) MEN1KMT2ADRD2DRD3SCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111601789-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 江苏凯迪恩医药科技有限公司 2020-08-28 CN disclosed
WO-2020124500-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏凯迪恩医药科技有限公司 2020-06-25 WO disclosed