SCHEMBL22129296

SCHEMBL22129296

COC(=O)C[C@@H](C)Nc1cc(Br)cc(F)c1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.38
MAPT P10636 5/20 0.38
PKM P14618 1/20 0.38
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 8/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GAA P10253 2/20 0.34
MAPK1 P28482 2/20 0.34
CASP6 P55212 1/20 0.33
RAB9A P51151 1/20 0.33
TNF P01375 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22129297 1.00 HCAR3 (0.38) HCAR3MAPTPKMMEN1KMT2A
SCHEMBL29743229 1.00 HCAR3 (0.38) HCAR3MAPTPKMMEN1KMT2A
SCHEMBL29743215 1.00 HCAR3 (0.38) HCAR3MAPTPKMMEN1KMT2A
SCHEMBL22129300 0.89 HCAR3 (0.39) HCAR3MAPTMEN1KMT2AALDH1A1
SCHEMBL22129301 0.89 HCAR3 (0.39) HCAR3MAPTMEN1KMT2AALDH1A1
SCHEMBL23749384 0.89 HCAR3 (0.39) HCAR3MAPTMEN1KMT2AALDH1A1
SCHEMBL18152724 0.85 HCAR3 (0.47) HCAR3MAPTPKMMEN1KMT2A
SCHEMBL21522752 0.84 HCAR3 (0.36) HCAR3MAPTPKMMEN1KMT2A
SCHEMBL22129298 0.82 ADRB2 (0.33) MAPTALDH1A1HTTSMN1; SMN2GAA
SCHEMBL22129305 0.82 ADRB2 (0.33) MAPTALDH1A1HTTSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020125513-A1 MACROCYCLIC COMPOUND AS CDK INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF IN MEDICINE 凯复制药有限公司 2020-06-25 WO disclosed