SCHEMBL2213201

SCHEMBL2213201

CN1CCCC1CCOc1ccc2nc(OC(=O)NCCC3CCOCC3)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.50
PDE3A Q14432 2/20 0.50
HRH3 Q9Y5N1 3/20 0.47
SCN9A Q15858 6/20 0.40
ATM Q13315 1/20 0.39
BRAF P15056 1/20 0.38
BRD4 O60885 1/20 0.37
POLR1A O95602 1/20 0.37
CHRM3 P20309 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1377383 0.88 PDE3B (0.52) PDE3BPDE3AHRH3SCN9A
SCHEMBL2209226 0.86 HRH3 (0.51) PDE3BPDE3AHRH3SCN9A
SCHEMBL2211917 0.83 HRH3 (0.46) PDE3BPDE3AHRH3ATMCHRM3
SCHEMBL2211145 0.78 HRH3 (0.58) HRH3
SCHEMBL2206296 0.77 HRH3 (0.52) HRH3
SCHEMBL1377269 0.76 HRH3 (0.59) PDE3BPDE3AHRH3SCN9A
SCHEMBL2209038 0.74 HRH3 (0.59) HRH3SCN9A
SCHEMBL2208645 0.74 HRH3 (0.58) PDE3BPDE3AHRH3SCN9AATM
SCHEMBL2211945 0.72 HRH3 (0.54) HRH3
SCHEMBL1377891 0.72 HRH3 (0.48) PDE3BPDE3AHRH3SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805166-B1 QUINOLINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-07-27 EP claimed