SCHEMBL22138697

SCHEMBL22138697

O=C(Nc1cnc2cc[nH]c2c1C1=C/C=C\C=C/C=C\1)C1CCCCCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
JAK3 P52333 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
RXFP2 Q8WXD0 1/20 0.36
CETP P11597 1/20 0.36
STK17B O94768 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
CDK2 P24941 2/20 0.35
CCNA2 P20248 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22138731 0.84 ROCK2 (0.44) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL19059708 0.81 HDAC3 (0.47) HDAC3HDAC1HDAC2ALDH1A1NPC1
SCHEMBL22853567 0.81 HDAC3 (0.47) HDAC3HDAC1HDAC2ALDH1A1NPC1
SCHEMBL21157257 0.80 RAB9A (0.43) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL20368588 0.77 HDAC3 (0.44) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL20368587 0.77 HDAC3 (0.44) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL21157773 0.77 HDAC3 (0.44) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL22018162 0.77 HDAC3 (0.44) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL22853729 0.77 CDK2 (0.41) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL22138688 0.76 HDAC3 (0.36) HDAC3HDAC1HDAC2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3670506-A1 THIAZOLECARBOXAMIDES AND PYRIDINECARBOXAMIDE COMPOUNDS USEFUL AS PIM KINASE INHIBITORS Incyte Holdings Corporation (US) 2020-06-24 EP disclosed