SCHEMBL2213895

SCHEMBL2213895

CC(Oc1ccc(Sc2ccc(Sc3nnc[nH]3)nc2C(=O)Nc2nc3cccnc3s2)cc1)N(C)C

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCK P35557 17/20 0.44
ADORA3 P0DMS8 1/20 0.33
BUB1 O43683 1/20 0.32
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2210566 0.88 GCK (0.44) GCK
SCHEMBL2211348 0.87 GCK (0.59) GCKNPC1RAB9A
SCHEMBL2211415 0.85 GCK (0.54) GCKNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2212536 0.84 GCK (0.52) GCKADORA3
SCHEMBL2211540 0.83 GCK (0.42) GCK
SCHEMBL2213440 0.79 GCK (0.38) GCKNPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2211357 0.79 GCK (0.55) GCKADORA3MEN1NPC1MAPT
SCHEMBL2215580 0.76 GCK (0.55) GCK
SCHEMBL2642911 0.75 GCK (0.75) GCKNPC1RAB9ASMN1; SMN2
SCHEMBL2211857 0.74 GCK (0.53) GCKMEN1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1598349-B1 NOVEL 2-PYRIDINECARBOXAMIDE DERIVATIVES MSD KK (JP) 2011-07-27 EP claimed