SCHEMBL22154694

SCHEMBL22154694

CCCCCCON(C(=O)[C@@H](N)[C@@H](C)CC)C(CC(O[Si](C)(C)C(C)(C)C)c1nc(C(=O)OCC)cs1)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.36
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
CA2 P00918 5/20 0.32
PLA2G4A P47712 1/20 0.32
CA12 O43570 4/20 0.32
CA1 P00915 4/20 0.32
CA9 Q16790 4/20 0.32
PTPRB P23467 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28633849 0.91 ABCB1 (0.35) ABCB1MEN1NPC1ALDH1A1MAPT
SCHEMBL28633853 0.91 ABCB1 (0.35) ABCB1MEN1NPC1ALDH1A1MAPT
SCHEMBL25829279 0.91 ABCB1 (0.35) ABCB1MEN1NPC1ALDH1A1MAPT
SCHEMBL25829278 0.88 ABCB1 (0.37) ABCB1MEN1NPC1ALDH1A1MAPT
SCHEMBL28632005 0.88 ABCB1 (0.34) ABCB1PLA2G4A
SCHEMBL28632004 0.88 ABCB1 (0.34) ABCB1PLA2G4A
SCHEMBL28631046 0.87 ABCB1 (0.43) ABCB1MEN1NPC1ALDH1A1MAPT
SCHEMBL28631048 0.87 ABCB1 (0.43) ABCB1MEN1NPC1ALDH1A1MAPT
SCHEMBL28627110 0.83 ABCB1 (0.33) ABCB1
SCHEMBL22154622 0.81 FAP (0.37) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020132658-A2 TUBULYSINS AND PROTEIN-TUBULYSIN CONJUGATES REGENERON PHARMACEUTICALS, INC. (US) 2020-06-25 WO disclosed