FAP
Prolyl endopeptidase FAP · Q12884 · FAP on Sugi Atlas →
63,343 patent compounds predicted against FAP, 31,280 high-confidence (nearest known ligand ≥ 0.5)
Top predicted compounds (top 20 by supporting neighbours, then confidence)
| Compound | Confidence | Supporting neighbours | |
|---|---|---|---|
| Dutogliptin (SCHEMBL164106) | 1.00 | 19/20 | |
| Talabostat (SCHEMBL393024) | 1.00 | 13/20 | |
| SCHEMBL301874 | 0.47 | 12/20 | |
| Denagliptin (SCHEMBL682185) | 0.67 | 10/20 | |
| Hydrochloric Acid (SCHEMBL295498) | 0.80 | 9/20 | |
| Hydrochloric Acid (SCHEMBL356162) | 0.80 | 9/20 | |
| SCHEMBL196303 | 0.61 | 9/20 | |
| SCHEMBL196304 | 0.61 | 9/20 | |
| SCHEMBL196984 | 0.61 | 9/20 | |
| SCHEMBL646728 | 0.47 | 9/20 | |
| SCHEMBL160189 | 0.53 | 7/20 | |
| SCHEMBL637987 | 0.49 | 7/20 | |
| SCHEMBL637493 | 0.71 | 6/20 | |
| SCHEMBL639988 | 0.71 | 6/20 | |
| SCHEMBL464681 | 0.55 | 6/20 | |
| Trifluoroacetic Acid (SCHEMBL572193) | 0.48 | 6/20 | |
| SCHEMBL636985 | 0.61 | 5/20 | |
| SCHEMBL639880 | 0.61 | 5/20 | |
| SCHEMBL639502 | 0.60 | 5/20 | |
| SCHEMBL554778 | 0.68 | 4/20 |
Clinical trials — most relevant to FAP by text similarity (a relevance ranking, not an exhaustive list)
Related proteins — ESM-2 sequence neighbours (a FAP binder may also engage these)
| Protein | Name | Similarity | |
|---|---|---|---|
| Q9Z218 | — | 1.000 | Q9Z218 → |
| P28843 | — | 1.000 | P28843 → |
| A5D7B7 | — | 1.000 | A5D7B7 → |
| P0DRB8 | — | 0.999 | P0DRB8 → |
| B2D0J4 | — | 0.999 | B2D0J4 → |
| B1A4F7 | — | 0.999 | B1A4F7 → |
| P42658 | — | 0.996 | P42658 → |
| P97321 | — | 0.996 | P97321 → |
| Q5IS50 | — | 0.996 | Q5IS50 → |
| P22411 | — | 0.995 | P22411 → |
| DPP4 | Dipeptidyl peptidase 4 | 0.995 | landscape → |
| O14073 | — | 0.995 | O14073 → |
| Q9N2I7 | — | 0.993 | Q9N2I7 → |
| Q18253 | — | 0.992 | Q18253 → |
| Q6NXK7 | — | 0.992 | Q6NXK7 → |
| P14740 | — | 0.992 | P14740 → |
| P81425 | — | 0.992 | P81425 → |
| B6V868 | — | 0.992 | B6V868 → |
| P18962 | — | 0.989 | P18962 → |
| Q8N608 | — | 0.989 | Q8N608 → |
| Q9P778 | — | 0.989 | Q9P778 → |
| P42659 | — | 0.988 | P42659 → |
| A1CHP1 | — | 0.988 | A1CHP1 → |
| P85841 | — | 0.988 | P85841 → |
| Q6Q629 | — | 0.987 | Q6Q629 → |
| A0A1Q3EPF5 | — | 0.987 | A0A1Q3EPF5 → |
| Q10916 | — | 0.987 | Q10916 → |
| P33894 | — | 0.986 | P33894 → |
| W4VSJ0 | — | 0.986 | W4VSJ0 → |
| Q9VTJ4 | — | 0.986 | Q9VTJ4 → |