SCHEMBL2215856

SCHEMBL2215856

Cc1cc(OCCCC2CCN(c3noc(C4CCCO4)n3)CC2)ccc1C(=O)N[C@H](C)CO

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AXL P30530 11/20 0.41
HRH3 Q9Y5N1 2/20 0.40
GPR119 Q8TDV5 2/20 0.37
RAF1 P04049 1/20 0.35
CNR2 P34972 2/20 0.35
CNR1 P21554 1/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2218058 1.00 AXL (0.41) AXLHRH3GPR119RAF1CNR2
SCHEMBL2215852 1.00 AXL (0.41) AXLHRH3GPR119RAF1CNR2
SCHEMBL1845766 0.90 GPR119 (0.39) AXLHRH3GPR119
SCHEMBL2214697 0.90 GPR119 (0.39) AXLHRH3GPR119
SCHEMBL2216051 0.90 GPR119 (0.39) AXLHRH3GPR119
SCHEMBL2216773 0.90 GPR119 (0.40) AXLHRH3GPR119
SCHEMBL2217649 0.89 HRH3 (0.37) AXLHRH3GPR119CNR2NPC1
SCHEMBL2217644 0.89 HRH3 (0.37) AXLHRH3GPR119CNR2NPC1
SCHEMBL2217652 0.88 GPR119 (0.38) AXLHRH3GPR119RAB9A
SCHEMBL13536459 0.88 GPR119 (0.39) AXLHRH3GPR119CNR2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110178054-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-07-21 US disclosed
US-20110178054-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-07-21 US disclosed
US-20110178054-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-07-21 US disclosed
WO-2010004348-A1 HETEROCYCLIC GPCR AGONISTS PROSIDION LIMITED (GB) 2010-01-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178054-A1 Heterocyclic GPCR Agonists GPR119, GCGR, GPR27 AXL 581/4885HRH3 406/4885GPR119 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.