SCHEMBL2216070

SCHEMBL2216070

Cc1cc(OCCCC2CCN(c3noc(C(C)(F)F)n3)CC2)ccc1C(=O)N[C@@H]1COC[C@H]1O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.42
ACACB O00763 4/20 0.40
ACACA Q13085 3/20 0.40
SCN9A Q15858 1/20 0.35
KCNH2 Q12809 2/20 0.34
TTK P33981 1/20 0.34
GPR84 Q9NQS5 1/20 0.33
CYP11B2 P19099 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TYK2 P29597 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2219840 1.00 GPR119 (0.42) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2215240 0.96 GPR119 (0.42) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2219251 0.96 GPR119 (0.42) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2216586 0.91 GPR119 (0.47) GPR119ACACBACACAKCNH2TTK
SCHEMBL2219780 0.91 GPR119 (0.44) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2217755 0.91 GPR119 (0.44) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2214693 0.88 GPR119 (0.48) GPR119ACACBACACAKCNH2TTK
SCHEMBL2217348 0.87 ACACB (0.45) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2216930 0.87 GPR119 (0.44) GPR119ACACBACACASCN9AKCNH2
SCHEMBL2217954 0.87 GPR119 (0.44) GPR119ACACBACACASCN9AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110178054-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-07-21 US disclosed
US-20110178054-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-07-21 US disclosed
US-20110178054-A1 Heterocyclic GPCR Agonists PROSIDION LIMITED (GB) 2011-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178054-A1 Heterocyclic GPCR Agonists GPR119, GCGR, GPR27 GPR119 1/4885ACACB 2654/4885ACACA 2114/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.