SCHEMBL221704

SCHEMBL221704

CC(=O)N(C)C(=O)N(C)C(C)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM3 P20309 1/20 0.38
LMNA P02545 2/20 0.36
TSHR P16473 3/20 0.33
ALDH1A1 P00352 2/20 0.33
THPO P40225 2/20 0.33
FFAR3 O14843 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33
PMP22 Q01453 2/20 0.31
CA1 P00915 1/20 0.31
ALOX15 P16050 1/20 0.31
BLM P54132 1/20 0.31
NFKB1 P19838 1/20 0.30
HSD17B10 Q99714 1/20 0.30
MAPT P10636 1/20 0.30
APEX1 P27695 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12957824 0.86 ALDH1A1 (0.37) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL21482179 0.85 LMNA (0.37) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL11731904 0.85 ALDH1A1 (0.45) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL992383 0.84
SCHEMBL16647104 0.81 CHRM2 (0.32) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL17532662 0.81 NQO1 (0.39)
SCHEMBL21486137 0.81 ALDH1A1 (0.36) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL21482175 0.76 TSHR (0.33) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL22644257 0.76 CHRM2 (0.30) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL22648830 0.76 CHRM2 (0.30) CHRM1CHRM2CHRM4CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105669479-B The method that one kettle way prepares the trans 4 dimethyl amido cronate hydrochlorate of high-purity 重庆威鹏药业有限公司 2018-04-13 CN claimed
EP-2272490-B1 Stabilization of body-care and household products against degradation by UV radiation using merocyanine derivatives BASF SE (DE) 2019-10-16 EP disclosed
US-20160370523-A1 POLARIZING PLATE COMPOSITION, POLARIZING PLATE PROTECTIVE FILM, POLARIZER, POLARIZING PLATE, AND LIQUID CRYSTAL DISPLAY DEVICE FUJIFILM CORPORATION (JP) 2016-12-22 US disclosed
EP-2588500-B1 COPOLYMERS OF MONOCARBOXYLIC ACIDS AND DICARBOXYLIC ACIDS, THEIR PREPARATION AND USE BASF SE (DE) 2016-08-10 EP disclosed
EP-2458989-B1 IN SITU PREPARATION OF PERACID-BASED REMOVABLE ANTIMICROBIAL COATING COMPOSITIONS AND METHODS OF USE DU PONT (US) 2013-10-09 EP disclosed
US-8497318-B2 Copolymers of monocarboxylic acids and dicarboxylic acids, their preparation and use BASF SE (DE) 2013-07-30 US disclosed
EP-2588500-A1 COPOLYMERS OF MONOCARBOXYLIC ACIDS AND DICARBOXYLIC ACIDS, THEIR PREPARATION AND USE BASF SE (DE) 2013-05-08 EP disclosed
EP-2458989-A2 IN SITU PREPARATION OF PERACID-BASED REMOVABLE ANTIMICROBIAL COATING COMPOSITIONS AND METHODS OF USE E. I. du Pont de Nemours and Company (US) 2012-06-06 EP disclosed
US-20120004383-A1 COPOLYMERS OF MONOCARBOXYLIC ACIDS AND DICARBOXYLIC ACIDS, THEIR PREPARATION AND USE BASF SE (DE) 2012-01-05 US disclosed
WO-2012001092-A1 COPOLYMERS OF MONOCARBOXYLIC ACIDS AND DICARBOXYLIC ACIDS, THEIR PREPARATION AND USE BASF SE (DE) 2012-01-05 WO disclosed
EP-0051987-B1 BLEACH ACTIVATOR COMPOSITIONS, PREPARATION THEREOF AND USE IN GRANULAR DETERGENT COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 1985-04-03 EP disclosed
EP-0034387-B1 MULLS CONTAINING CHAIN STRUCTURE CLAY SUSPENSION AIDS THE PROCTER & GAMBLE COMPANY (US) 1984-10-24 EP disclosed
US-4444674-A Granular bleach activator compositions and detergent compositions containing them THE PROCTER & GAMBLE COMPANY (US) 1984-04-24 US disclosed
EP-0028432-B1 GRANULAR LAUNDRY COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 1984-01-18 EP disclosed
US-4399049-A PARTICLES EXTRUDED WITH ETHOXYLATED NONIONIC SURFACTANT; STORAGE STABILITY; RABID DISPERSION; LAUNDERING THE PROCTER & GAMBLE COMPANY (US) 1983-08-16 US disclosed
US-4321157-A SILICA OR SILICATE, ORGANIC PEROXY ACID BLEACH PRECURSOR, ALIPHATIC ALCOHOL-ALKYLENE OXIDE CONDENSATE NONIONIC SURFACTANT THE PROCTER & GAMBLE COMPANY (US) 1982-03-23 US disclosed
EP-0034387-A2 Mulls containing chain structure clay suspension aids THE PROCTER & GAMBLE COMPANY (US) 1981-08-26 EP disclosed
US-4264466-A LAUNDRY DETERGENTS THE PROCTER & GAMBLE COMPANY (US) 1981-04-28 US disclosed
US-4248928-A TETRAACETYL AKYLENEDIAMINES OR TETRAACETYL GLYCOURIL PEROXY BLEACH PRECURSOR THE PROCTER & GAMBLE COMPANY (US) 1981-02-03 US disclosed
US-4179390-A Laundry additive product THE PROCTER & GAMBLE COMPANY (US) 1979-12-18 US disclosed