SCHEMBL22174993

SCHEMBL22174993

C=CC(=O)N1CCN(c2ccc(C)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.59
LMNA P02545 3/20 0.55
ACHE P22303 2/20 0.51
MAPT P10636 4/20 0.50
ALDH1A1 P00352 3/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
HTT P42858 1/20 0.50
GAA P10253 2/20 0.49
GFER P55789 2/20 0.49
POLB P06746 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALOX15 P16050 1/20 0.49
ALOX12 P18054 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KIT P10721 1/20 0.48
AURKB Q96GD4 1/20 0.48
CASP6 P55212 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20456544 0.83 MAPT (0.63) LMNAMAPTALDH1A1POLBKDM4E
SCHEMBL29773303 0.83 GFER (0.65) AKR1C3LMNAMAPTALDH1A1CYP2C9
SCHEMBL21583811 0.83 AKR1C3 (0.61) AKR1C3LMNAMAPTALDH1A1HPGD
SCHEMBL8014611 0.82 ALDH1A1 (0.61) AKR1C3LMNAMAPTALDH1A1CYP2C9
SCHEMBL24267460 0.82 PANK3 (0.54) LMNAMAPTALDH1A1HPGDHTT
SCHEMBL25787603 0.82 MAPT (0.61) LMNAMAPTALDH1A1HTTGAA
SCHEMBL25045164 0.82 MAPT (0.56) LMNAMAPTALDH1A1HTTGAA
SCHEMBL20456543 0.82 L3MBTL1 (0.68) AKR1C3ACHEMAPTALDH1A1HTT
Toluene SCHEMBL28499348 0.80 KMT2A (0.57) ACHEMAPTALDH1A1HTTPOLB
SCHEMBL630856 0.80 AKR1C3 (0.65) AKR1C3LMNAMAPTALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3805214-B1 JAK3 SELECTIVE INHIBITOR UNIV PEKING SHENZHEN GRADUATE SCHOOL (CN) 2023-07-05 EP disclosed
EP-3805214-A1 JAK3 SELECTIVE INHIBITOR Peking University Shenzhen Graduate School (CN) 2021-04-14 EP disclosed
WO-2020140055-A1 CYCLIN-DEPENDENT KINASE INHIBITORS SPV THERAPEUTICS INC. (US) 2020-07-02 WO disclosed
WO-2020140054-A1 CYCLIN-DEPENDENT KINASE INHIBITORS SPV THERAPEUTICS INC. (US) 2020-07-02 WO disclosed