SCHEMBL2218201

SCHEMBL2218201

CCCCc1nc(C(=O)O)cc2c3ccccc3n(Cc3ccccc3)c12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.47
AGTR2 P50052 6/20 0.47
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.46
PDE4C Q08493 3/20 0.46
PDE4D Q08499 3/20 0.46
TLR7 Q9NYK1 3/20 0.43
CYP19A1 P11511 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
FOLH1 Q04609 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2212262 0.93 PDE4A (0.48) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL28273846 0.93 CYP19A1 (0.47) CYP19A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL28273845 0.93 CYP19A1 (0.47) CYP19A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL28273840 0.92 CYP19A1 (0.46) AGTR1AGTR2CYP19A1KDM4ECYP1A2
SCHEMBL2215730 0.90 ALDH1A1 (0.43) KDM4E
SCHEMBL2216828 0.89 PGR (0.46) KDM4E
SCHEMBL2214735 0.89 CYP19A1 (0.47) CYP19A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL28273849 0.88 KDM4E (0.52) AGTR1AGTR2KDM4EHSD17B10
SCHEMBL28273854 0.88 KDM4E (0.52) AGTR1AGTR2KDM4EHSD17B10
SCHEMBL28869106 0.87 KDM4E (0.51) AGTR1AGTR2KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1634881-B1 HARMINE DERIVATIVES, INTERMEDIATES USED IN THEIR PREPARATION, PREPARATION PROCESSES AND USE THEREOF XINJIANG HUASHIDAN PHARMACEUTICAL RES CO LTD (CN) 2011-07-27 EP claimed