SCHEMBL22198962

SCHEMBL22198962

Cc1cc2ccc(F)c(Cl)c2[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.43
RIPK1 Q13546 1/20 0.43
BRD4 O60885 13/20 0.42
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
DAO P14920 3/20 0.40
ATAD2 Q6PL18 11/20 0.39
DDO Q99489 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22185211 0.81 TNF (0.41) TNFRIPK1GRIN2DGRIN3BGRIN1
SCHEMBL3363264 0.80 DAO (0.61) TNFRIPK1GRIN2DGRIN3BGRIN1
SCHEMBL22184937 0.80 EIF4A3 (0.40) TNFRIPK1GRIN2DGRIN3BGRIN1
SCHEMBL22198970 0.78 HRH4 (0.45) BRD4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL22198968 0.78 NQO2 (0.43) BRD4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12970395 0.76 DAO (0.65) BRD4DAOATAD2DDO
SCHEMBL25310064 0.73 BRD4 (0.42) BRD4DAOATAD2DDO
SCHEMBL30482258 0.73 BRD4 (0.42) BRD4DAOATAD2DDO
SCHEMBL25262124 0.73 PARP1 (0.44) BRD4DAOATAD2DDO
SCHEMBL30482246 0.73 PARP1 (0.44) BRD4DAOATAD2DDO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed