SCHEMBL22199024

SCHEMBL22199024

Cc1cn(-c2ccncc2)cn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.62
CYP2A6 P11509 1/20 0.62
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP19A1 P11511 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
MAPK13 O15264 1/20 0.43
NR2E1 Q9Y466 2/20 0.42
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
MAOA P21397 3/20 0.40
MAOB P27338 3/20 0.40
WNT3A P56704 1/20 0.39
EGLN2 Q96KS0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27985278 0.87 CYP1A2 (0.65) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL2283022 0.81 CYP2E1 (0.65) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL22199099 0.79 CYP2E1 (0.62) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL18754697 0.78 CYP3A4 (0.56) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL19272800 0.78 CYP1A2 (0.56) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL242918 0.78 CYP2E1 (0.51) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL4668245 0.78 CYP1A2 (0.56) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL12988609 0.78 CYP3A4 (0.56) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL4666728 0.78 CYP3A4 (0.56) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6
SCHEMBL22198914 0.77 NR2E1 (0.60) CYP2E1CYP2A6CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed