SCHEMBL22199029

SCHEMBL22199029

Cc1cn(-c2ccccn2)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.52
CYP2E1 P05181 1/20 0.50
CYP2A6 P11509 1/20 0.50
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
PLD1 Q13393 1/20 0.42
CPB1 P15086 1/20 0.41
CPB2 Q96IY4 1/20 0.41
KDM4E B2RXH2 2/20 0.41
POLB P06746 1/20 0.41
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
GRM5 P41594 1/20 0.40
SLC11A2 P49281 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27966806 0.86 EGLN2 (0.55) EGLN2SMN1; SMN2CYP2E1CYP2A6CPB1
SCHEMBL22184926 0.78 CYP2E1 (0.51) EGLN2SMN1; SMN2CYP2E1CYP2A6KDM4E
SCHEMBL31095576 0.77 NOS3 (0.45) EGLN2SMN1; SMN2ALDH1A1HTTHSD17B10
SCHEMBL13177332 0.77 KDM4E (0.64) EGLN2SMN1; SMN2CYP2E1CYP2A6ALDH1A1
SCHEMBL6172976 0.77 SMN1; SMN2 (0.43) EGLN2SMN1; SMN2ALDH1A1HTTHSD17B10
SCHEMBL2159955 0.77 NOS3 (0.45) EGLN2SMN1; SMN2ALDH1A1HTTHSD17B10
SCHEMBL30337851 0.77 SMN1; SMN2 (0.43) EGLN2SMN1; SMN2ALDH1A1HTTHSD17B10
SCHEMBL12759471 0.77 SMN1; SMN2 (0.43) EGLN2SMN1; SMN2ALDH1A1HTTHSD17B10
SCHEMBL22185839 0.77 CPB2 (0.44) EGLN2SMN1; SMN2ALDH1A1HTTHSD17B10
SCHEMBL4752191 0.76 EGLN2 (1.00) EGLN2SMN1; SMN2KDM4ESLC11A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed