SCHEMBL22199044

SCHEMBL22199044

COc1ccc(Oc2ccc(C)cc2C)cc1C

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.52
GAA P10253 1/20 0.48
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 1/20 0.47
AR P10275 7/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
SLC6A4 P31645 3/20 0.41
HTR2A P28223 2/20 0.41
KCNH2 Q12809 2/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303786 0.86 ACHE (0.54) ACHEGAAALDH1A1CYP3A4AR
SCHEMBL12248268 0.86 SLC6A4 (0.46) ACHEGAAL3MBTL1SLC6A4HTR2A
SCHEMBL25620294 0.86 CA12 (0.50) ACHEALDH1A1CYP3A4ARL3MBTL1
SCHEMBL28452075 0.86 SLC6A4 (0.45) ACHEGAAALDH1A1ARL3MBTL1
SCHEMBL144308 0.85 ACHE (0.68) ACHEGAAALDH1A1CYP3A4L3MBTL1
SCHEMBL29352952 0.85 ACHE (0.68) ACHEGAAALDH1A1CYP3A4L3MBTL1
SCHEMBL446449 0.84 AR (0.47) ACHEGAAALDH1A1ARL3MBTL1
Ammonia Solution, Strong SCHEMBL6473680 0.83 ACHE (0.65) ACHEGAAALDH1A1CYP3A4L3MBTL1
SCHEMBL13011575 0.82 TEAD4 (0.50) ACHEALDH1A1ARL3MBTL1SLC6A4
SCHEMBL11767346 0.81 CA12 (0.59) ACHEGAAALDH1A1CYP3A4AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed