SCHEMBL22200426

SCHEMBL22200426

COC(=O)CCC(F)(F)c1cc2cc3c(cc2s1)OCO3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RAB9A P51151 9/20 0.38
ALDH1A1 P00352 4/20 0.38
NPC1 O15118 8/20 0.38
SMN1; SMN2 Q16637 5/20 0.38
KDM4E B2RXH2 8/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
MAPT P10636 4/20 0.36
NPSR1 Q6W5P4 2/20 0.36
NFKB1 P19838 1/20 0.36
PPARG P37231 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
NCOA2 Q15596 1/20 0.36
NCOA1 Q15788 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200413 0.93 SMN1; SMN2 (0.45) MEN1KMT2ARAB9AALDH1A1NPC1
SCHEMBL22200397 0.85 NPC1 (0.36) MEN1KMT2ARAB9AALDH1A1NPC1
SCHEMBL22200286 0.80 STING1 (0.49)
SCHEMBL22200406 0.78 ALDH1A1 (0.40) MEN1KMT2ARAB9AALDH1A1NPC1
SCHEMBL22200423 0.78 STING1 (0.50) MEN1KMT2ARAB9AALDH1A1
SCHEMBL24175827 0.77 STING1 (0.45)
SCHEMBL22200623 0.76 STING1 (0.51)
SCHEMBL22200624 0.74 STING1 (0.54)
SCHEMBL24175175 0.73 ACHE (0.43)
SCHEMBL24175161 0.70 STING1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3907221-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2021-11-10 EP disclosed
WO-2020140894-A1 FLUORINE-CONTAINING SUBSTITUTED BENZOTHIOPHENE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 中国科学院上海药物研究所 2020-07-09 WO disclosed