SCHEMBL22211534

SCHEMBL22211534

Nc1ccc(Cl)cc1-c1cc(C(F)(F)P)ncn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.42
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KMO O15229 1/20 0.35
DYRK3 O43781 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35
DYRK2 Q92630 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
CYP3A4 P08684 2/20 0.34
TSHR P16473 2/20 0.34
ALOX15 P16050 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CA2 P00918 1/20 0.33
CHKA P35790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16068268 0.88 CA2 (0.46) IDO1ALDH1A1KDM4EHSD17B10KMO
SCHEMBL22211420 0.83 MPL (0.37) ALDH1A1KDM4EHSD17B10CA2CHKA
SCHEMBL22211794 0.83 IDO1 (0.42) IDO1KDM4ECA2CHKAPIM3
SCHEMBL18700477 0.77 IDO1 (0.47) IDO1ALDH1A1HSD17B10KMODYRK3
SCHEMBL39774 0.77 IDO1 (0.50) IDO1ALDH1A1KMODYRK3CCNA2
SCHEMBL22211510 0.74 IDO1 (0.42) IDO1ALDH1A1KDM4EHSD17B10DYRK3
SCHEMBL17392797 0.72 CA2 (0.47) ALDH1A1KDM4EHSD17B10CA2CHKA
SCHEMBL16971331 0.71 IDO1 (0.44) IDO1ALDH1A1KDM4EDYRK3CCNA2
SCHEMBL16068058 0.71 CA2 (0.46) IDO1ALDH1A1KDM4EHSD17B10KMO
SCHEMBL16068170 0.71 AGPAT2 (0.44) IDO1ALDH1A1KDM4EHSD17B10KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975030-B1 DIHYDROPYRIDAZINE-3,5-DIONE DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 2020-07-15 EP disclosed