SCHEMBL2221172

SCHEMBL2221172

CO[C@@H](C)CN(C)c1cnc(C(N)=O)cn1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.45
ACACB O00763 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
TSHR P16473 1/20 0.33
MC4R P32245 1/20 0.33
ADRA1A P35348 1/20 0.33
MC3R P41968 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
HCAR3 P49019 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
FPR2 P25090 1/20 0.31
SCN9A Q15858 1/20 0.31
NNMT P40261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037386 0.80 SIRT6 (0.41) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL30482977 0.77 SIRT6 (0.46) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL2793061 0.77 SIRT6 (0.47) SIRT6ADRA1AHCAR3HSP90AA1HSP90AB1
SCHEMBL30874243 0.77 SIRT6 (0.52) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL2222631 0.77 SIRT6 (0.52) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL30301027 0.74 SIRT6 (0.46) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL5042470 0.72 HCAR3 (0.46) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL5132655 0.70 RPS6KB1 (0.46) SIRT6
SCHEMBL5133491 0.70 HCAR3 (0.43) SIRT6TSHRHCAR3
SCHEMBL5042293 0.68 SIRT6 (0.40) SIRT6ADORA3TSHRMC4RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed