SCHEMBL22213404

SCHEMBL22213404

CN(N)/C(Cc1ncc(N)c(-c2ccccc2)n1)=N\N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 1/20 0.35
SKP1 P63208 1/20 0.35
SKP2 Q13309 1/20 0.35
MAPT P10636 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ADK P55263 4/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NR4A2 P43354 1/20 0.32
NUDT1 P36639 2/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18779303 0.73 ALDH1A1 (0.46) CKS1BSKP1SKP2MAPTADORA2A
SCHEMBL17111687 0.73 ALDH1A1 (0.46) MAPTKMT2ACYP1A2HPGDHTT
SCHEMBL18779357 0.72 CYP1A2 (0.40) MAPTMEN1KMT2AADORA2AADORA1
SCHEMBL18792160 0.72 DPP4 (0.45) MAPTL3MBTL1MEN1KMT2AADORA2A
SCHEMBL17111581 0.72 PTGS2 (0.40) MAPTL3MBTL1ADORA2AADORA1HPGD
SCHEMBL17110527 0.69 CKS1B (0.38) CKS1BSKP1SKP2MAPTADK
SCHEMBL16585346 0.68 MAPT (0.54) CKS1BSKP1SKP2MAPTL3MBTL1
Hydrochloric Acid SCHEMBL16585666 0.67 MAPT (0.53) CKS1BSKP1SKP2MAPTL3MBTL1
SCHEMBL17111663 0.67 SRC (0.40) MAPTMEN1KMT2AADORA2AADORA1
SCHEMBL17111479 0.67 NTRK1 (0.40) MAPTMEN1KMT2AADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3122346-B1 TRKA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME (US) 2020-07-15 EP disclosed