SCHEMBL22216353

SCHEMBL22216353

COC(=O)c1cnn(C/C(=C/F)CN2C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 5/20 0.42
MAPT P10636 3/20 0.42
NPC1 O15118 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
GAA P10253 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29441565 1.00 POLB (0.51) POLBMAPK1HSD17B10ALDH1A1MAPT
SCHEMBL23907174 0.86 KMT2A (0.45) POLBALDH1A1MAPTNPSR1KDM4E
SCHEMBL23907175 0.86 KMT2A (0.45) POLBALDH1A1MAPTNPSR1KDM4E
SCHEMBL23920594 0.86 ALDH1A1 (0.51) POLBMAPK1ALDH1A1MAPTNPC1
SCHEMBL22216351 0.83 KDM4E (0.37) POLBHSD17B10ALDH1A1NPSR1KDM4E
SCHEMBL22206964 0.80 KMT2A (0.47) POLBMAPK1HSD17B10ALDH1A1MAPT
SCHEMBL22206965 0.80 KMT2A (0.47) POLBMAPK1HSD17B10ALDH1A1MAPT
SCHEMBL28427551 0.80 POLB (0.53) POLBMAPK1HSD17B10ALDH1A1MAPT
SCHEMBL22216441 0.80 POLB (0.53) POLBMAPK1HSD17B10ALDH1A1MAPT
SCHEMBL29441569 0.80 POLB (0.53) POLBMAPK1HSD17B10ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892621-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF Nanjing Transthera Biosciences Co., Ltd. (CN) 2021-10-13 EP disclosed
WO-2020143763-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF 南京药捷安康生物科技有限公司 2020-07-16 WO disclosed