SCHEMBL2222137

SCHEMBL2222137

OCCc1cnc(-c2cccc(Cl)c2)nc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 6/20 0.56
HRH1 P35367 1/20 0.44
IDO1 P14902 2/20 0.42
MAOB P27338 2/20 0.42
TAAR1 Q96RJ0 1/20 0.42
ADORA1 P30542 2/20 0.42
FYN P06241 1/20 0.41
HIF1A Q16665 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2223578 0.88 FYN (0.48) PDE4BHRH1IDO1TAAR1FYN
SCHEMBL2220568 0.81 PDE4B (0.42) PDE4BHRH1IDO1MAOBTAAR1
SCHEMBL13273284 0.81 PDE4B (0.50) PDE4BHRH1IDO1TAAR1LMNA
SCHEMBL2269848 0.78 PDE4B (0.45) PDE4BIDO1TAAR1LMNAPOLB
SCHEMBL2220953 0.78 NR1I3 (0.43) PDE4BHRH1IDO1TAAR1LMNA
SCHEMBL2616114 0.75 IDO1 (0.47) IDO1LMNAPOLBMAPT
SCHEMBL2131570 0.75 DHFR (0.51) HRH1IDO1MAOBADORA1
SCHEMBL9250325 0.75 MAOB (0.46) HRH1IDO1MAOBTAAR1HIF1A
SCHEMBL13275140 0.75 NPC1 (0.55) POLBGAAMAPT
SCHEMBL2557747 0.75 IDO1 (0.44) HRH1IDO1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2515657-A1 TYROSINE KINASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-10-31 EP disclosed
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed