SCHEMBL9250325

SCHEMBL9250325

C=CCCc1cnc(-c2ccc(-c3cccc(Cl)c3)cc2)nc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.46
TAAR1 Q96RJ0 2/20 0.45
HRH1 P35367 1/20 0.38
PGR P06401 2/20 0.37
ALOX5 P09917 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
HIF1A Q16665 1/20 0.36
SLC6A7 Q99884 1/20 0.36
IDO1 P14902 1/20 0.36
MAP4K4 O95819 3/20 0.36
USP1 O94782 1/20 0.35
WDR48 Q8TAF3 1/20 0.35
CNR2 P34972 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252692 0.84 SMN1; SMN2 (0.37) MAOBKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9252364 0.81 CYP11B1 (0.41) HSD17B10
SCHEMBL9252963 0.77 RARB (0.40) MAOBKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9253788 0.76 RARB (0.40) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2222137 0.75 PDE4B (0.56) MAOBTAAR1HRH1HIF1AIDO1
SCHEMBL9406468 0.75 RARB (0.36) MAOBKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9249705 0.74 CYP11B1 (0.36) HSD17B10
SCHEMBL9406670 0.74 RARB (0.41) TAAR1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9251920 0.73 CYP11B1 (0.39) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9131495 0.72 TAAR1 (0.57) TAAR1ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5454974-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1995-10-03 US disclosed
US-5302317-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-04-12 US disclosed
EP-0315014-B1 Halogenated benzene derivatives HOFFMANN LA ROCHE (CH) 1994-01-12 EP disclosed
US-5230826-A HALOBENZENE LIQUID CRYSTALS HOFFMANN-LA ROCHE INC. (US) 1993-07-27 US disclosed
EP-0315014-A2 Halogenated benzene derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed