SCHEMBL2222743

SCHEMBL2222743

O=C(O)c1c(-c2ccccc2)ccnc1N1CCN(Cc2cccc(OCc3ccccc3)c2)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.58
LMNA P02545 4/20 0.58
ALDH1A1 P00352 4/20 0.58
HTT P42858 3/20 0.58
TSHR P16473 2/20 0.58
HPGD P15428 1/20 0.58
ALOX12 P18054 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
FAAH O00519 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.48
CD274 Q9NZQ7 1/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALOX15 P16050 1/20 0.46
GAA P10253 1/20 0.46
DRD2 P14416 2/20 0.45
DRD4 P21917 2/20 0.45
DRD3 P35462 2/20 0.45
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2222893 0.89 KDM4E (0.52) KDM4ELMNAALDH1A1HTTTSHR
SCHEMBL2225912 0.80 CD274 (0.47) KDM4ELMNAALDH1A1HTTTSHR
SCHEMBL2223195 0.80 KDM4E (0.47) KDM4ELMNAALDH1A1HTTTSHR
SCHEMBL2225112 0.79 KDM4E (0.49) KDM4ELMNAALDH1A1HTTTSHR
SCHEMBL14554261 0.79 NPC1 (0.50) KDM4ELMNAALDH1A1HTTSMN1; SMN2
SCHEMBL15678972 0.76 MAPT (0.42) KDM4ELMNAL3MBTL1MEN1KMT2A
SCHEMBL14554258 0.76 KDM4E (0.44) KDM4ELMNAALDH1A1HTTTSHR
SCHEMBL2223087 0.76 MEN1 (0.47) KDM4ELMNAALDH1A1HTTTSHR
SCHEMBL2222903 0.75 HTR3E (0.47) KDM4ELMNAALDH1A1HTTHPGD
Hydrochloric Acid SCHEMBL2225347 0.75 MEN1 (0.47) KDM4ELMNAALDH1A1HTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523665-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS Glaxo Group Limited (GB) 2012-11-21 EP disclosed
WO-2011088201-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS GLAXO GROUP LIMITED (GB) 2011-07-21 WO disclosed