SCHEMBL22229656

SCHEMBL22229656

Cc1cc(C)c(-c2cc3ccccc3c(-c3c(O)c(-c4c(C)cc(C)cc4C)cc4ccccc34)c2O)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.53
CYP2A6 P11509 1/20 0.53
NQO1 P15559 1/20 0.42
GPR84 Q9NQS5 4/20 0.41
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
ALOX5 P09917 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 1/20 0.38
TRPM4 Q8TD43 1/20 0.37
PKM P14618 1/20 0.37
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
KDM4E B2RXH2 1/20 0.36
THRB P10828 1/20 0.36
NQO2 P16083 1/20 0.36
CRHR1 P34998 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31388613 1.00 CYP1A2 (0.53) CYP1A2CYP2A6NQO1GPR84LMNA
SCHEMBL14327814 0.89 CYP1A2 (0.46) CYP1A2CYP2A6NQO1GPR84MEN1
SCHEMBL14327813 0.88 CYP1A2 (0.52) CYP1A2CYP2A6NQO1GPR84LMNA
SCHEMBL3927495 0.88 CYP1A2 (0.45) CYP1A2CYP2A6NQO1GPR84LMNA
SCHEMBL19159038 0.85 CYP1A2 (0.42) CYP1A2CYP2A6NQO1GPR84ALOX5
SCHEMBL18575590 0.83 GPR84 (0.44) CYP1A2CYP2A6NQO1GPR84ALOX5
SCHEMBL7098784 0.81 ALOX5 (0.50) CYP1A2NQO1GPR84ALOX5MEN1
SCHEMBL29514619 0.81 ALOX5 (0.50) CYP1A2NQO1GPR84ALOX5MEN1
SCHEMBL25485142 0.81 NQO1 (0.44) CYP1A2CYP2A6NQO1GPR84LMNA
SCHEMBL22229714 0.79 GPR84 (0.58) CYP1A2CYP2A6NQO1GPR84ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11664093-B2 Extrapolative prediction of enantioselectivity enabled by computer-driven workflow, new molecular representations and machine learning THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-30 US disclosed
US-20200234798-A1 EXTRAPOLATIVE PREDICTION OF ENANTIOSELECTIVITY ENABLED BY COMPUTER-DRIVEN WORKFLOW, NEW MOLECULAR REPRESENTATIONS AND MACHINE LEARNING THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2020-07-23 US disclosed