SCHEMBL22230481

SCHEMBL22230481

CC(=O)Nc1cncc(-c2ccc(C)c(NS(=O)(=O)c3ccc(F)c(F)c3)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
CYP2C9 P11712 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PIK3C3 Q8NEB9 3/20 0.46
BDKRB1 P46663 1/20 0.46
PIP4K2A P48426 2/20 0.44
PIP4K2B P78356 2/20 0.44
AKT1 P31749 4/20 0.43
PIK3CA P42336 4/20 0.43
MTOR P42345 4/20 0.43
PKM P14618 2/20 0.43
PRF1 P14222 1/20 0.42
PIK3CB P42338 2/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CG P48736 1/20 0.41
PRKDC P78527 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28800820 0.90 PKM (0.52) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL28946371 0.88 AKT1 (0.52) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL28800837 0.88 TSHR (0.53) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL28800826 0.86 ACLY (0.47) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL29808034 0.85 TP53 (0.54) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL22230460 0.85 TP53 (0.54) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL28800816 0.85 AKT1 (0.54) TP53MAPTSMN1; SMN2PIK3C3BDKRB1
SCHEMBL22230480 0.85 PIP4K2A (0.50) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL28800815 0.84 PIK3C3 (0.58) TSHRCYP2C9TP53MAPTSMN1; SMN2
SCHEMBL28800806 0.83 PIK3C3 (0.56) PIK3C3PIK3CAPRF1PIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109721531-B Novel liposome kinase inhibitor 中国科学院合肥物质科学研究院 2022-07-29 CN disclosed
WO-2020147097-A1 NOVEL LIPOSOME KINASE INHIBITOR 中国科学院合肥物质科学研究院 2020-07-23 WO disclosed