SCHEMBL2223911

SCHEMBL2223911

CO[C@H](C)CN(C)c1cnc(C(=O)NCc2ccc3c(c2)CCN(C2CCC2)CC3)cn1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 16/20 0.49
HRH1 P35367 1/20 0.47
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2D6 P10635 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269194 1.00 HRH3 (0.49) HRH3HRH1ALDH1A1CYP1A2POLB
SCHEMBL2267296 0.89 HRH3 (0.51) HRH3HRH1LMNA
SCHEMBL2266798 0.89 HRH3 (0.51) HRH3HRH1LMNA
SCHEMBL2264332 0.89 HRH3 (0.54) HRH3HRH1ALDH1A1CYP1A2POLB
SCHEMBL2191302 0.86 HRH3 (0.48) HRH3HRH1CYP2D6
SCHEMBL2191319 0.86 HRH3 (0.48) HRH3HRH1CYP2D6
SCHEMBL1789991 0.80 HRH3 (0.51) HRH3HRH1
SCHEMBL1789988 0.80 HRH3 (0.51) HRH3HRH1
SCHEMBL1791368 0.80 HRH3 (0.51) HRH3HRH1
SCHEMBL2275230 0.79 HRH3 (0.55) HRH3HRH1ALDH1A1CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO claimed
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed