SCHEMBL2267296

SCHEMBL2267296

CO[C@@H](C)CN(C)c1ccc(C(=O)NCc2ccc3c(c2)CCN(C2CCC2)CC3)cn1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.51
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
HRH1 P35367 1/20 0.40
ADRA1A P35348 1/20 0.38
MAPK14 Q16539 1/20 0.38
CXCR3 P49682 1/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2266798 1.00 HRH3 (0.51) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL1789991 0.91 HRH3 (0.51) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL1789988 0.91 HRH3 (0.51) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL1791368 0.91 HRH3 (0.51) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL2191319 0.91 HRH3 (0.48) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL2191302 0.91 HRH3 (0.48) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL2269194 0.89 HRH3 (0.49) HRH3HRH1LMNA
SCHEMBL2223911 0.89 HRH3 (0.49) HRH3HRH1LMNA
SCHEMBL1789947 0.89 HRH3 (0.52) HRH3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL2268812 0.88 ADRA1A (0.51) HRH3PRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed
WO-2011083315-A1 COMPOUNDS AND THEIR USE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed