SCHEMBL22239228

SCHEMBL22239228

Nc1ccc(C(=O)Cl)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA13 Q8N1Q1 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
P4HA1 P13674 1/20 0.38
MIF P14174 1/20 0.38
P4HTM Q9NXG6 1/20 0.38
HIF1A Q16665 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249720 0.80 P4HTM (0.59) P4HA1MIFP4HTMHIF1AKDM4E
SCHEMBL31359466 0.80 P4HTM (0.59) P4HA1MIFP4HTMHIF1AKDM4E
SCHEMBL1831265 0.80 KMT2A (0.55) SIRT6CA12CA1CA2CA4
SCHEMBL27212642 0.79 P2RX7 (0.52) HIF1AKDM4EALDH1A1MAOBPTGS1
SCHEMBL26697541 0.79 HDAC1 (0.47) HIF1AKDM4EALDH1A1MAOBPTGS1
SCHEMBL30753596 0.78 ALDH1A1 (0.47) CA12CA1CA2CA4CA6
Hydrochloric Acid SCHEMBL21485420 0.78 P4HTM (0.57) ADRA2AADRA2BADRA2CP4HA1MIF
SCHEMBL28015545 0.78 ALDH1A1 (0.47) CA12CA1CA2CA4CA6
SCHEMBL19470150 0.78 CA12 (0.41) CA12CA1CA2CA4CA6
SCHEMBL995902 0.78 ALDH1A1 (0.47) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3683207-A1 N-ALKYLARYL-5-OXYARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B Cadent Therapeutics, Inc. (US) 2020-07-22 EP disclosed