SCHEMBL22248293

SCHEMBL22248293

NC1CC2(CCN(Cc3ccc(-n4ccc(NC(=O)N5CCNCC5)nc4=O)cc3)CC2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.36
KDM1A O60341 1/20 0.35
MAOB P27338 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35
HPGD P15428 1/20 0.34
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
MEN1 O00255 3/20 0.33
CYP2C9 P11712 3/20 0.33
KMT2A Q03164 3/20 0.33
CYP3A4 P08684 3/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP2C19 P33261 2/20 0.33
TSHR P16473 2/20 0.33
HIF1A Q16665 2/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
IKBKE Q14164 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22248413 0.92 HPGD (0.36) ROCK2KDM1AMAOBRCOR1HPGD
SCHEMBL22248888 0.92 HTR2A (0.33) ROCK2KCNH2CYP2D6CYP1A2
SCHEMBL22248665 0.91 KDM1A (0.37) KDM1AMAOBRCOR1HPGDHDAC3
SCHEMBL22248357 0.91 ROCK2 (0.35) ROCK2IKBKETBK1FAAH
SCHEMBL22248664 0.90 HPGD (0.44) KDM1AMAOBRCOR1HPGDHDAC3
SCHEMBL22248670 0.90 FAAH (0.36) ROCK2CYP2D6CYP1A2FAAH
SCHEMBL22235832 0.89 ROCK2 (0.35) ROCK2KDM1AMAOBRCOR1HPGD
SCHEMBL22248295 0.89 ROCK2 (0.38) ROCK2FAAH
SCHEMBL22254537 0.88 ROCK2 (0.39) ROCK2FAAH
SCHEMBL22248411 0.87 CXCR4 (0.39) MEN1KMT2AFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150372-A1 ANTIMICROBIAL COMPOUNDS AND METHODS CURZA GLOBAL, LLC (US) 2020-07-23 WO disclosed