SCHEMBL2225550

SCHEMBL2225550

Cc1cc(-c2nc3cnc(Oc4cncc(Cl)c4)nc3o2)cc(C)c1[O]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.56
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
PPARG P37231 1/20 0.32
CYP1A2 P05177 8/20 0.32
CYP3A4 P08684 7/20 0.32
USP2 O75604 5/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
CYP2C9 P11712 6/20 0.32
ALDH1A1 P00352 5/20 0.32
TSHR P16473 5/20 0.32
CYP2C19 P33261 4/20 0.32
HSD17B10 Q99714 3/20 0.32
MAPK1 P28482 2/20 0.32
CYP2D6 P10635 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
CASP1 P29466 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2224638 0.89 S1PR1 (0.48) S1PR1TP53ALDH1A1HSD17B10
SCHEMBL2224494 0.87 S1PR1 (0.47) S1PR1CYP1A2CYP3A4USP2TP53
SCHEMBL2222853 0.87 S1PR1 (0.58) S1PR1GAAHTTCYP1A2CYP3A4
SCHEMBL2223355 0.86 S1PR1 (0.73) S1PR1CYP1A2CYP3A4USP2LMNA
SCHEMBL2222499 0.85 S1PR1 (0.54) S1PR1CYP1A2CYP3A4USP2LMNA
SCHEMBL14797179 0.85 S1PR1 (0.79) S1PR1HTTPPARGCYP1A2CYP3A4
SCHEMBL2224653 0.83 S1PR1 (0.56) S1PR1PPARGCYP1A2CYP3A4USP2
SCHEMBL2222343 0.82 S1PR1 (0.56) S1PR1CYP1A2CYP3A4USP2LMNA
SCHEMBL2227168 0.82 S1PR1 (0.52) S1PR1HTTCYP1A2CYP3A4USP2
SCHEMBL2222401 0.81 S1PR1 (0.49) S1PR1CYP1A2CYP3A4USP2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523962-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI (FR) 2012-11-21 EP disclosed
WO-2011086079-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI-AVENTIS (FR) 2011-07-21 WO disclosed