SCHEMBL22256294

SCHEMBL22256294

OC1=C(c2c(O)c(-c3ccc(C4CCCCC4)cc3)cc3c2CCCC3)C2=C(CCCC2)CC1c1ccc(C2CCCCC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 1/20 0.30
APP P05067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25195073 0.82 KMT2A (0.54) MEN1KMT2ACYP3A4CYP2C9APP
SCHEMBL22256347 0.76 CYP3A4 (0.32) CYP3A4CYP2C9APP
SCHEMBL22256292 0.68 TGFBR1 (0.38) MEN1KMT2ACYP3A4CYP2C9APP
SCHEMBL22229749 0.67 CYP3A4 (0.40) MEN1KMT2ACYP3A4CYP2C9APP
SCHEMBL16772616 0.63 MEN1 (0.64) MEN1KMT2A
SCHEMBL4127678 0.61 MEN1 (0.56) MEN1KMT2AAPP
SCHEMBL1044154 0.59 MEN1 (0.38) MEN1KMT2A
SCHEMBL4123679 0.59 KMT2A (0.54) MEN1KMT2A
SCHEMBL9000030 0.58 NUDT1 (0.38) KMT2ACYP3A4CYP2C9APP
SCHEMBL3919336 0.57 MEN1 (0.51) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11664093-B2 Extrapolative prediction of enantioselectivity enabled by computer-driven workflow, new molecular representations and machine learning THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-30 US disclosed
US-20200234798-A1 EXTRAPOLATIVE PREDICTION OF ENANTIOSELECTIVITY ENABLED BY COMPUTER-DRIVEN WORKFLOW, NEW MOLECULAR REPRESENTATIONS AND MACHINE LEARNING THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2020-07-23 US disclosed