SCHEMBL22258772

SCHEMBL22258772

CN(C)c1ccnc(C(=O)Nc2c[nH]nc2-c2ccccn2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 5/20 0.41
GAA P10253 4/20 0.41
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CYP3A4 P08684 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
GFER P55789 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13314759 0.79 MCL1 (0.54) ALDH1A1MAPTNPC1RAB9ACYP3A4
SCHEMBL3579872 0.76 ALDH1A1 (0.47) ALDH1A1KDM4EMAPTGAANPC1
SCHEMBL20086026 0.75 IRAK4 (0.48) MAPTGAANPC1RAB9ANPSR1
SCHEMBL13314750 0.75 NPC1 (0.49) ALDH1A1MAPTGAANPC1RAB9A
SCHEMBL13314755 0.73 JAK2 (0.44) MAPTNPC1RAB9APOLBLMNA
Formic Acid SCHEMBL29911871 0.72 IRAK4 (0.46) MAPTGAANPC1RAB9ANPSR1
SCHEMBL23719268 0.71 ADORA3 (0.51) MAPTNPC1RAB9ALMNAKMT2A
SCHEMBL18170033 0.71 CHEK1 (0.55) NPC1RAB9ATLR7
SCHEMBL29752180 0.71 CHEK1 (0.55) NPC1RAB9ATLR7
SCHEMBL20415626 0.69 TLR7 (0.36) ALDH1A1KDM4EMAPTGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed