SCHEMBL2226163

SCHEMBL2226163

CCC(C)C(C(=O)O)N1Cc2ccc(-c3ccc(NC(=O)c4ccc(-c5ccccc5)cc4)cc3C(F)(F)F)cc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.45
ATM Q13315 1/20 0.45
ALDH1A1 P00352 1/20 0.44
PKM P14618 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
ITGB3 P05106 2/20 0.42
ITGA2B P08514 2/20 0.42
ITGA2 P17301 2/20 0.42
S1PR1 P21453 14/20 0.42
S1PR3 Q99500 7/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13718844 0.92 S1PR1 (0.44) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL2224457 0.92 S1PR1 (0.44) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL2178689 0.87 S1PR1 (0.44) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL2365141 0.86 AKR1C3 (0.46) GAAATMALDH1A1PKMMAPK1
SCHEMBL2178623 0.85 ITGB3 (0.42) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL2178629 0.85 ITGB3 (0.42) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL13719612 0.84 AKR1C3 (0.44) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL2181367 0.84 AKR1C3 (0.44) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL13718848 0.83 PLK1 (0.41) ITGB3ITGA2BITGA2S1PR1S1PR3
SCHEMBL2177053 0.83 MEN1 (0.45) ALDH1A1ITGB3ITGA2BITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2519500-A1 INHIBITORS OF DIACYLGLYCEROL ACYL TRANSFERASE Piramal Healthcare Ltd. (IN) 2012-11-07 EP disclosed
WO-2011080718-A1 INHIBITORS OF DIACYLGLYCEROL ACYL TRANSFERASE PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-07-07 WO disclosed