SCHEMBL2226596

SCHEMBL2226596

O=Cc1ccc(CCc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
CYP2A6 P11509 2/20 0.59
MAOA P21397 3/20 0.50
MAOB P27338 3/20 0.50
FFAR1 O14842 1/20 0.50
RAB9A P51151 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
ALOX12 P18054 1/20 0.44
CASP1 P29466 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HDAC1 Q13547 2/20 0.44
CALM1 P0DP23 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
KEAP1 Q14145 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
HTR2A P28223 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14369268 1.00 ALDH1A1 (0.59) ALDH1A1CYP2A6MAOAMAOBFFAR1
SCHEMBL17278365 0.91 ALDH1A1 (0.54) ALDH1A1CYP2A6MAOAMAOBALOX15
SCHEMBL2225297 0.91 ALDH1A1 (0.54) ALDH1A1CYP2A6MAOAMAOBHDAC1
SCHEMBL5429778 0.90 CYP2A6 (0.50) ALDH1A1CYP2A6RAB9AHPGDHSD17B10
SCHEMBL2222928 0.88 ALDH1A1 (0.62) ALDH1A1CYP2A6MAOAMAOBRAB9A
Tannin Pyrogallol SCHEMBL28930134 0.85 ALDH1A1 (0.58) ALDH1A1CYP2A6MAOAMAOBFFAR1
SCHEMBL14330452 0.83 CYP2A6 (0.44) ALDH1A1CYP2A6RAB9AHPGDHSD17B10
SCHEMBL9371806 0.82 CYP1A2 (0.56) ALDH1A1CYP2A6MAOAMAOBRAB9A
SCHEMBL2323602 0.82 HDAC8 (0.59) ALDH1A1CYP2A6MAOAHDAC1TDP1
SCHEMBL6494686 0.82 ALDH1A1 (0.48) ALDH1A1CYP2A6MAOAMAOBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4582903-A Synthesis of unsaturated hydantoins with an inexpensive catalyst STAUFFER CHEMICAL COMPANY (US) 1986-04-15 US claimed
US-4345072-A Process for the production of 5-arylidene hydantoins (B) DEGUSSA AG (DE) 1982-08-17 US claimed
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed
EP-2692717-B1 METHOD FOR PRODUCING 4,4'-DIFORMYLDIPHENYLALKANE MITSUBISHI GAS CHEMICAL CO (JP) 2015-05-13 EP disclosed
US-8969627-B2 Method for producing 4,4'-diformyldiphenylalkane MITSUBISHI GAS CHEMICAL COMPANY, INC (JP) 2015-03-03 US disclosed
US-8841327-B2 Heterocycles substituted pyridine derivatives and antifungal agent containing thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2014-09-23 US disclosed
EP-2692717-A1 METHOD FOR PRODUCING 4,4'-DIFORMYLDIPHENYLALKANE Mitsubishi Gas Chemical Company, Inc. (JP) 2014-02-05 EP disclosed
US-20130023541-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS GLAXO GROUP LIMITED 2013-01-24 US disclosed
CN-102802627-A Voltage-gated sodium channel blockers GLAXO GROUP LTD 2012-11-28 CN disclosed
EP-2523665-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS Glaxo Group Limited (GB) 2012-11-21 EP disclosed
US-3954833-A PROSTAGLANDINS THE UPJOHN COMPANY (US) 1976-05-04 US disclosed
US-3944595-A PROSTAGLANDIN THE UPJOHN COMPANY (US) 1976-03-16 US disclosed
US-3933898-A ANTIULCER, ANTICOAGULANTS, NASAL PATENCY, LABOR INDUCERS, WOUND HEALING THE UPJOHN COMPANY (US) 1976-01-20 US disclosed
US-3933895-A PROSTAGLANDINS, ANTIULCER, ANTICOAGULANTS, NASAL PATENCY, LABOR INDUCERS, WOUND HEALING THE UPJOHN COMPANY (US) 1976-01-20 US disclosed
US-3933897-A ANTIULCER, ASTHMA, RENAL DYSFUNCTION THE UPJOHN COMPANY (US) 1976-01-20 US disclosed
US-3933896-A ANTICOAGULANTS, ASTHMA, LABOR INDUCERS, CERVICAL DILATION THE UPJOHN COMPANY (US) 1976-01-20 US disclosed
US-3933900-A ANTIULCER, ANTICOAGULANTS, NASAL PATENCY, LABOR INDUCERS, WOUND HEALING THE UPJOHN COMPANY (US) 1976-01-20 US disclosed
US-3933899-A ANTIULCER, ANTICOAGULANTS, NASAL PATENCY, LABOR INDUCERS, WOUND HEALING THE UPJOHN COMPANY (US) 1976-01-20 US disclosed
US-3931279-A 5-Oxa prostaglandin F2.sub.α analogs THE UPJOHN COMPANY (US) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130023541-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS KCNB1, KCNB2, SCNN1B ALDH1A1 2656/4885CYP2A6 2295/4885MAOA 1655/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.