SCHEMBL2226673

SCHEMBL2226673

Cc1cc([C@@H]2CNC[C@]2(CN)Cc2ccccc2)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.41
SLC6A3 Q01959 5/20 0.41
KCNH2 Q12809 2/20 0.41
KDM1A O60341 7/20 0.36
RCOR1 Q9UKL0 3/20 0.36
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35
SLC6A4 P31645 5/20 0.33
CYP2D6 P10635 2/20 0.32
MAOA P21397 6/20 0.32
MAOB P27338 6/20 0.32
TRPM4 Q8TD43 1/20 0.31
TRPM5 Q9NZQ8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228602 0.91 SLC6A2 (0.41) SLC6A2SLC6A3KCNH2KDM1ARCOR1
SCHEMBL2225309 0.90 SLC6A2 (0.39) SLC6A2SLC6A3KCNH2KDM1ARCOR1
SCHEMBL2228579 0.90 SLC6A2 (0.39) SLC6A2SLC6A3KCNH2KDM1ARCOR1
SCHEMBL2228553 0.90 SLC6A2 (0.39) SLC6A2SLC6A3KCNH2KDM1ARCOR1
SCHEMBL2225021 0.83 KDM1A (0.52) SLC6A2SLC6A3KDM1ARCOR1SLC6A4
SCHEMBL1421527 0.83 KDM1A (0.52) SLC6A2SLC6A3KDM1ARCOR1SLC6A4
SCHEMBL3634310 0.81 MAOA (0.47) KDM1ARCOR1MAOAMAOB
SCHEMBL2352598 0.78 KDM1A (0.52) SLC6A2SLC6A3KDM1ARCOR1OPRM1
SCHEMBL2228338 0.78 KDM1A (0.52) SLC6A2SLC6A3KDM1ARCOR1OPRM1
SCHEMBL2784188 0.78 SLC6A2 (0.39) SLC6A2SLC6A3KCNH2SLC6A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513052-A1 PYRROLIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011085886-A1 PYRROLIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-07-21 WO disclosed