SCHEMBL22275943

SCHEMBL22275943

Cn1nc(-c2cccc(OCCCn3nc(-c4ccc(Cl)s4)c4c(N)ncnc43)c2)c2c(N)ncnc21

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 16/20 0.50
PRKDC P78527 16/20 0.50
PIK3CA P42336 15/20 0.50
PIK3CB P42338 15/20 0.50
PIK3CG P48736 15/20 0.50
SRC P12931 11/20 0.48
ABL1 P00519 10/20 0.48
EGFR P00533 9/20 0.48
HCK P08631 9/20 0.48
MTOR P42345 9/20 0.48
EPHB4 P54760 9/20 0.48
KDR P35968 9/20 0.48
NUDT14 O95848 1/20 0.46
NUDT5 Q9UKK9 1/20 0.46
PI4KB Q9UBF8 3/20 0.46
RET P07949 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24157345 0.88 KDR (0.41) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL129539 0.79 PIK3CD (0.59) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL130468 0.79 PIK3CD (0.65) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL129870 0.76 SRC (0.77) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL130590 0.74 SRC (0.73) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL128513 0.73 PIK3CD (0.67) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL17970673 0.71 PIK3CD (0.65) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL197491 0.71 PIK3CD (0.65) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL22275941 0.70 PIK3CD (0.51) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG
SCHEMBL12351 0.70 PIK3CD (0.74) PIK3CDPRKDCPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200239427-A1 NOVEL KINASE MODULATORS RHIZEN PHARMACEUTICALS AG (CH) 2020-07-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200239427-A1 NOVEL KINASE MODULATORS PRKCA, PRKCH, PRKCB PIK3CD 70/4885PRKDC 164/4885PIK3CA 143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.