SCHEMBL22280426

SCHEMBL22280426

COC(=O)c1cccc(-c2cnco2)c1OC

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 16/20 0.46
IMPDH1 P20839 4/20 0.46
EDNRA P25101 1/20 0.45
AAK1 Q2M2I8 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14840095 0.86 KDM4E (0.52) IMPDH2EDNRAAAK1
SCHEMBL22280594 0.84 EDNRA (0.45) IMPDH2IMPDH1EDNRAAAK1
SCHEMBL22280423 0.76 FAAH (0.43)
SCHEMBL24026537 0.76 IMPDH2 (0.43) IMPDH2IMPDH1AAK1
SCHEMBL24026459 0.76 IMPDH2 (0.44) IMPDH2IMPDH1AAK1
SCHEMBL7723821 0.76 IMPDH2 (0.47) IMPDH2IMPDH1AAK1
SCHEMBL21376047 0.76 IMPDH2 (0.52) IMPDH2IMPDH1AAK1
SCHEMBL24720275 0.76 IMPDH2 (0.46) IMPDH2IMPDH1AAK1
SCHEMBL30930931 0.76 IMPDH2 (0.46) IMPDH2IMPDH1AAK1
SCHEMBL20150098 0.74 AAK1 (0.46) IMPDH2IMPDH1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020153431-A1 ESTER COMPOUND 第一三共株式会社 2020-07-30 WO disclosed
WO-2020153431-A1 ESTER COMPOUND 第一三共株式会社 2020-07-30 WO disclosed