SCHEMBL22280459

SCHEMBL22280459

Cc1ccc(Nc2ccc(C#N)cn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
CYP2A6 P11509 1/20 0.48
CSNK1A1 P48729 1/20 0.48
CSNK1D P48730 1/20 0.48
GSK3B P49841 1/20 0.48
CSNK1G2 P78368 1/20 0.48
CCR6 P51684 1/20 0.46
SLC2A1 P11166 1/20 0.46
TRPV4 Q9HBA0 1/20 0.45
MAPKAPK2 P49137 1/20 0.45
GRM5 P41594 1/20 0.44
HAO1 Q9UJM8 1/20 0.44
ABCG2 Q9UNQ0 3/20 0.43
KDM4E B2RXH2 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 1/20 0.42
DHODH Q02127 1/20 0.42
CDK1 P06493 1/20 0.42
KDR P35968 1/20 0.42
CCNK O75909 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27303096 0.84 GRM5 (0.46) ALDH1A1CYP2A6CCR6TRPV4GRM5
SCHEMBL27295837 0.83 MEN1 (0.51) TRPV4GRM5ABCG2DHODHLMNA
SCHEMBL31473409 0.83 MEN1 (0.51) TRPV4GRM5ABCG2DHODHLMNA
SCHEMBL10549553 0.83 ABCG2 (0.53) ALDH1A1GSK3BABCG2KDM4EGAA
SCHEMBL11563207 0.80 HAO1 (0.53) GRM5HAO1KDR
SCHEMBL22265881 0.78 HPGD (0.53) ALDH1A1ABCG2KDM4EL3MBTL1LMNA
SCHEMBL10694580 0.78 ALDH1A1 (0.73) ALDH1A1CYP2A6CSNK1A1CSNK1DGSK3B
SCHEMBL22265747 0.76 HSD17B10 (0.56) ALDH1A1ABCG2KDM4EL3MBTL1GAA
SCHEMBL27297664 0.76 IDH1 (0.42) SLC2A1TRPV4ABCG2CCNKCCNA2
SCHEMBL27834535 0.75 CCNK (0.55) CSNK1A1CSNK1DCSNK1G2CCNKCCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020154431-A1 INHIBITORS OF SPINSTER HOMOLOG 2 (SPNS2) FOR USE IN THERAPY LYNCH KEVIN R (US) 2020-07-30 WO disclosed