SCHEMBL22280564

SCHEMBL22280564

Cc1ccc(-c2noc(C[C@@H]3CCNC3)n2)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.47
PLAT P00750 1/20 0.47
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
TLR9 Q9NR96 2/20 0.40
TLR8 Q9NR97 2/20 0.40
TLR7 Q9NYK1 2/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.39
HDAC4 P56524 3/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KIT P10721 1/20 0.38
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22280507 0.87 CNR1 (0.46) S1PR1PLATCNR1CNR2TLR9
Hydrochloric Acid SCHEMBL29523302 0.83 SPHK1 (0.41) TLR9TLR8TLR7
SCHEMBL22280458 0.81 ALDH1A1 (0.54) RAB9AALDH1A1TSHRRECQLNPC1
SCHEMBL22280454 0.81 ALDH1A1 (0.54) RAB9AALDH1A1TSHRRECQLNPC1
SCHEMBL22280455 0.76 TLR9 (0.50) S1PR1PLATTLR9TLR8TLR7
SCHEMBL22280440 0.74 ALDH1A1 (0.55) RAB9AALDH1A1TSHRRECQLNPC1
SCHEMBL22280635 0.74 S1PR1 (0.54) S1PR1PLATTLR9TLR8TLR7
SCHEMBL21387529 0.72 KIT (0.49) PLATCNR1CNR2TLR9TLR8
SCHEMBL12267064 0.71 S1PR1 (0.66) S1PR1PLATHDAC6LMNA
SCHEMBL22280647 0.71 S1PR1 (0.53) S1PR1PLATRAB9ATSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020154431-A1 INHIBITORS OF SPINSTER HOMOLOG 2 (SPNS2) FOR USE IN THERAPY LYNCH KEVIN R (US) 2020-07-30 WO disclosed