SCHEMBL22280802

SCHEMBL22280802

N#Cc1cccc2c1CCOC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.37
NOTUM Q6P988 2/20 0.34
PNMT P11086 1/20 0.34
DRD2 P14416 1/20 0.33
TSHR P16473 1/20 0.32
HSD11B1 P28845 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
MAPK1 P28482 1/20 0.31
CASP1 P29466 1/20 0.31
CYP2C19 P33261 1/20 0.31
HBB P68871 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30173200 0.76 NOTUM (0.44) TRPA1NOTUMPNMTDRD2TSHR
SCHEMBL4092520 0.75 HTR2A (0.54) HSD11B1MAPK1
SCHEMBL31394006 0.73 ABHD6 (0.33) TRPA1PNMT
SCHEMBL9120020 0.73 AKR1C3 (0.31)
SCHEMBL30817469 0.73 BCL2L1 (0.53) DRD2CA1CA2
SCHEMBL1597761 0.73 BCL2L1 (0.53) DRD2CA1CA2
SCHEMBL10615520 0.73 PARP1 (0.37) NOTUMKDM4EALDH1A1CYP1A2
SCHEMBL19835774 0.73 ADRA2A (0.47) PNMTHSD11B1
SCHEMBL5363757 0.73 ABHD6 (0.33) TRPA1PNMT
SCHEMBL26130065 0.73 CD44 (0.47) DRD2TSHRKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020153431-A1 ESTER COMPOUND 第一三共株式会社 2020-07-30 WO disclosed
WO-2020153431-A1 ESTER COMPOUND 第一三共株式会社 2020-07-30 WO disclosed