SCHEMBL2228404

SCHEMBL2228404

CC(C)N=Cc1c(NC(C)C)nc2ccccn2c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
NPSR1 Q6W5P4 3/20 0.54
HPGD P15428 2/20 0.54
ALOX15 P16050 1/20 0.54
KDM4E B2RXH2 5/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
LMNA P02545 1/20 0.49
USP7 Q93009 1/20 0.47
MAPT P10636 4/20 0.44
NPC1 O15118 1/20 0.40
ADORA1 P30542 1/20 0.40
HTT P42858 1/20 0.40
HCRTR1 O43613 1/20 0.40
POLB P06746 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GAA P10253 2/20 0.39
RAB9A P51151 1/20 0.39
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12517343 1.00 ALDH1A1 (0.54) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL3955431 0.77 USP7 (0.53) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL3960626 0.71 USP7 (0.53) ALDH1A1NPSR1KDM4EUSP7MAPT
SCHEMBL12517344 0.70 KDM4E (0.59) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL2229210 0.70 KDM4E (0.59) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL12517349 0.68 ALDH1A1 (0.78) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL2228146 0.68 ALDH1A1 (0.78) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL12517342 0.68 KDM4E (0.60) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL2227307 0.68 KDM4E (0.60) ALDH1A1NPSR1HPGDALOX15KDM4E
SCHEMBL12517662 0.68 ALDH1A1 (0.50) ALDH1A1NPSR1HPGDALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011089457-A1 NOVEL MEDICINAL COMPOUNDS URATIM GYÁRTÓ KORLÁTOLT FELELŐSSÉGŰ TÁRSASÁG (HU) 2011-07-28 WO claimed
WO-2011089457-A1 NOVEL MEDICINAL COMPOUNDS URATIM GYÁRTÓ KORLÁTOLT FELELŐSSÉGŰ TÁRSASÁG (HU) 2011-07-28 WO disclosed