SCHEMBL2228606

SCHEMBL2228606

CNC1CN(Cc2ccccc2)CC1c1ccc(C)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.44
CCR5 P51681 4/20 0.43
DPP4 P27487 1/20 0.42
RORC P51449 1/20 0.41
SCN4A P35499 2/20 0.39
SIGMAR1 Q99720 1/20 0.39
POLB P06746 2/20 0.38
LMNA P02545 1/20 0.38
DRD2 P14416 3/20 0.38
DRD3 P35462 3/20 0.38
DRD4 P21917 2/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1977456 1.00 KDM1A (0.44) KDM1ACCR5DPP4RORCSCN4A
SCHEMBL1974966 0.90 DPP4 (0.42) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL2226675 0.90 DPP4 (0.42) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL1974894 0.90 SIGMAR1 (0.47) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL2225316 0.90 SIGMAR1 (0.47) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL1974850 0.90 SIGMAR1 (0.47) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL1976032 0.90 SIGMAR1 (0.47) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL2413984 0.84 DPP4 (0.41) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL1975962 0.83 RORC (0.48) KDM1ACCR5DPP4RORCSIGMAR1
SCHEMBL1203069 0.83 RORC (0.48) KDM1ACCR5DPP4RORCSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513052-A1 PYRROLIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011085886-A1 PYRROLIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-07-21 WO disclosed