SCHEMBL22288679

SCHEMBL22288679

COCC1OC2(CCN(C(=O)O)CC2)CN(C)C1=O

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 19/20 0.49
OPRM1 P35372 17/20 0.49
KCNH2 Q12809 12/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17317227 0.82 SIGMAR1 (0.45) SIGMAR1OPRM1KCNH2
SCHEMBL17317160 0.81 SIGMAR1 (0.43) SIGMAR1OPRM1KCNH2
SCHEMBL20555604 0.80 SIGMAR1 (0.56) SIGMAR1OPRM1KCNH2
SCHEMBL17324904 0.73 OPRM1 (0.51) SIGMAR1OPRM1KCNH2
SCHEMBL19518142 0.73 OPRM1 (0.51) SIGMAR1OPRM1KCNH2
SCHEMBL20555587 0.69 SIGMAR1 (0.53) SIGMAR1OPRM1KCNH2
SCHEMBL12492762 0.69 OPRM1 (0.34) SIGMAR1OPRM1KCNH2
SCHEMBL19518229 0.69 OPRM1 (0.37) SIGMAR1OPRM1KCNH2
SCHEMBL20504475 0.68 SIGMAR1 (0.59) SIGMAR1OPRM1KCNH2
SCHEMBL17317132 0.68 OPRM1 (0.42) SIGMAR1OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020157026-A1 HYDROXYLATED DERIVATIVES OF 1-OXA-4,9-DIAZASPIRO UNDECANE COMPOUNDS HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-08-06 WO disclosed