SCHEMBL2229695

SCHEMBL2229695

CSCC[C@H](N)C(=O)OC(=O)[C@@H](N)Cc1c[nH]c2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSC P53634 4/20 0.63
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
KDM4E B2RXH2 2/20 0.58
MAPT P10636 2/20 0.58
LMNA P02545 1/20 0.58
MPO P05164 1/20 0.58
TSHR P16473 1/20 0.58
BLM P54132 1/20 0.58
PMP22 Q01453 1/20 0.58
HIF1A Q16665 1/20 0.58
TACR1 P25103 2/20 0.57
HTR2A P28223 2/20 0.50
ADRB1 P08588 1/20 0.50
HTR1A P08908 1/20 0.50
ADRA2A P08913 1/20 0.50
SLC6A2 P23975 1/20 0.50
HTR1D P28221 1/20 0.50
HTR1B P28222 1/20 0.50
HTR2C P28335 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3421789 0.90 CTSC (0.60) CTSCMEN1KMT2AKDM4EMAPT
SCHEMBL475351 0.88 MAPT (0.74) MEN1KMT2AKDM4EMAPTLMNA
SCHEMBL289044 0.88 MAPT (0.74) MEN1KMT2AKDM4EMAPTLMNA
Dl-Tryptophan SCHEMBL11461241 0.86 KMT2A (0.76) CTSCMEN1KMT2AKDM4EMAPT
Tryptophan SCHEMBL2229691 0.86 KMT2A (0.76) CTSCMEN1KMT2AKDM4EMAPT
Dl-Tryptophan SCHEMBL23924440 0.86 KMT2A (0.76) CTSCMEN1KMT2AKDM4EMAPT
Dl-Tryptophan SCHEMBL2229687 0.86 KMT2A (0.76) CTSCMEN1KMT2AKDM4EMAPT
SCHEMBL5065255 0.84 KDM4E (0.65) CTSCMEN1KMT2AKDM4EMAPT
Methionine SCHEMBL8860166 0.84 MEN1 (0.49) CTSCMEN1KMT2AKDM4EMAPT
SCHEMBL3401965 0.84 KDM4E (0.64) MEN1KMT2AKDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024131837-A1 ENGINEERED NUCLEASE WITH HIGH SALT TOLERANCE WUXI BIOLOGICS (SHANGHAI) CO., LTD. (CN) 2024-06-27 WO claimed
WO-2020069862-A1 PREPARATION OF AMINO ACIDS FROM THEIR AMINO NITRILES EVONIK OPERATIONS GMBH (DE) 2020-04-09 WO claimed
WO-2020069859-A1 SALT-FREE PREPARATION OF AMINO ACIDS FROM THEIR AMINO NITRILES EVONIK OPERATIONS GMBH (DE) 2020-04-09 WO claimed
EP-3632895-A1 SALT-FREE PRODUCTION OF AMINO ACIDS FROM THEIR AMINONITRILES Evonik Operations GmbH (DE) 2020-04-08 EP claimed
EP-3632896-A1 PRODUCTION OF AMINO ACIDS FROM THEIR AMINONITRILES Evonik Operations GmbH (DE) 2020-04-08 EP claimed
WO-2024131837-A1 ENGINEERED NUCLEASE WITH HIGH SALT TOLERANCE WUXI BIOLOGICS (SHANGHAI) CO., LTD. (CN) 2024-06-27 WO disclosed
US-20240093248-A1 CELLS AND METHOD OF CELL CULTURE PFIZER INC. (US) 2024-03-21 US disclosed
US-11718864-B2 Cells and method of cell culture PFIZER INC. (US) 2023-08-08 US disclosed
WO-2023126510-A1 MONOOXYGENASE MUTANTS FOR BIOSYNTHESIS OF 2,6-BIS(HYDROXYMETHYL)PYRIDINE AND A METHOD FOR PREPARATION OF 2,6-BIS(HYDROXYMETHYL)PYRIDINE USING THE SAID MONOOXYGENASE MUTANTS VIO CHEMICALS AG (CH) 2023-07-06 WO disclosed
US-20220386649-A1 COMPOSITION COMPRISING AMINO ACIDS AND A LIPID MATRIX FOR NON-MAMMALIAN MONOGASTRIC ANIMALS AND USE THEREOF VETAGRO INTERNATIONAL S.R.L. (IT) 2022-12-08 US disclosed
EP-4003051-A1 GRANULAR COMPOSITION COMPRISING AMINO ACIDS AND PHYTOCOMPOUNDS EMBEDDED IN A LIPID MATRIX FOR NON-MAMMALIAN MONOGASTRIC ANIMALS AND USE THEREOF Vetagro International S.r.l. (IT) 2022-06-01 EP disclosed
US-10947596-B2 Compositions and methods for identification, assessment, prevention, and treatment of cancer using NFS1 biomarkers and modulators DANA-FARBER CANCER INSTITUTE, INC. (US) 2021-03-16 US disclosed
WO-1999047173-A2 CARRIER FOR IN VIVO DELIVERY OF A THERAPEUTIC AGENT UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 1999-09-23 WO disclosed
WO-1999015662-A9 TELOMERE REPEAT BINDING FACTORS AND DIAGNOSTIC AND THERAPEUTIC USE THEREOF UNIV ROCKEFELLER (US) 1999-07-08 WO disclosed
WO-1999021995-A1 TREATMENT AND PREVENTION OF NEURODEGENERATIVE DISEASES USING MODULATORS OF THE INTERACTION OF APP AND A POLYPEPTIDE DEFINING A PI DOMAIN THE ROCKEFELLER UNIVERSITY (US) 1999-05-06 WO disclosed
WO-1999015662-A1 TELOMERE REPEAT BINDING FACTORS AND DIAGNOSTIC AND THERAPEUTIC USE THEREOF THE ROCKEFELLER UNIVERSITY (US) 1999-04-01 WO disclosed
WO-1999009056-A1 INHIBITION OF HIV-1 REPLICATION USING D-AMINO ACID PEPTIDES UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 1999-02-25 WO disclosed
WO-1999009199-A2 ELONGATION FACTOR-2 KINASE (EF-2 KINASE) AND METHODS OF USE THEREFOR UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 1999-02-25 WO disclosed
CN-1161001-A Lipid metabolism-improving agent KYOWA HAKKO KOGYO KK (JP) 1997-10-01 CN disclosed
US-5559142-A NUTRIENTS JAROWSKI CHARLES I (US) 1996-09-24 US disclosed